Table 1.
Mouse pharmacokinetic parameters after 8 mg/kg i.p. administration of ketamine.
Cmax (ng/mL) | V (L) | AUCinf (ng.h/L) | t1/2,α (h) | t1/2,β (h) | CLd (L/h) | CL (L/h) | B/P ratio | |
---|---|---|---|---|---|---|---|---|
P15 | 463 ± 87 | 115 ± 38 | 122 ± 26 | 0.05 ± 0.03 | 0.28 ± 0.17 | 157 ± 78 | 71 ± 12 | 14.7 ± 1 |
P30 | 1760 ± 231 | 81 ± 12 | 296 ± 48 | 0.09 ± 0.03 | 0.25 ± 0.13 | 284 ± 86 | 30 ± 7.2 | 8.7 ± 3.7 |
Adults | 1209 ± 152.5 | 69 ± 4 | 366 ± 59 | 0.07 ± 0.01 | 1.11 ± 0.8 | 326 ± 51 | 48 ± 3 | 2.7 ± 0.5 |
Cmax : maximum concentration, V: volume of distribution, AUCinf: area under the concentration time curve (AUC) with the last concentration extrapolated based on the elimination rate constant, t1/2,α: distribution of half-life, t1/2,β: elimination half-life, CLd: distribution clearance, CL: systemic clearance, B/P: brain to plasma ratio. Data are expressed as mean ± SEM.