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IC50 values of bisubstrate compounds
| Compound ID | IC50 (nM)a |
|---|---|
| 1 (NAH-C2-GPKRIA) | 260±70 |
| 2 (NAH-C3-GPKRIA) | 130±40 |
| 3 (NAH-C4-GPKRIA) | 82±17 |
| 4 (NAH-C5-GPKRIA) | N.A. |
| 5 (NAH-C2-GPKR) | 320±80 |
| 6 (NAH-C3-GPKR) | 200±30 |
| 7 (NAH-C4-GPKR) | 84±12 |
triplicates (n = 3). N.A.: not applied.
