Table 6.
Coupling of Benzoxazolyl Thioglycosides to 1,2;3,4-Di-O-isopropylidenegalactopyranose with Activation by Cu(OTf)2 in CH2Cl2 at Room Temperaturea
Entry | Donor | Product, % yield, β:α ratio |
---|---|---|
1 | ![]() |
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2 | ![]() |
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3 | ![]() |
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4 | ![]() |
No reactio (95% recovered donor) |
ROH = 1,2;3,4-di-O-ispropylidene-α-D-galactopyranose