Table 7.
XR | Activator |
---|---|
O-(Benz-1,3-oxazol-2-yl) | Cu(OTf)2 and DMTST |
O-5-pentenyl | IDCP, but not NIS, NBS, or NIS/TfOH |
S-Et | MeOTf, DMTST, I2, but not IDCP |
S-Ph and S-tolyl | I2, no significant difference |
S-(1,3-thiazolin-2-yl) | I2, no significant difference |