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. Author manuscript; available in PMC: 2020 Aug 17.
Published in final edited form as: J Med Chem. 2019 Feb 26;62(5):2666–2689. doi: 10.1021/acs.jmedchem.8b02008

Table 3.

Permeability Values of 12a and 7

# PAMPA Papp (cm/s) PAMPA–BBB Papp (cm/s)
12a (EML741)   4.8 × 10−7   2.3 × 10−7
7 (UNC0638)   0.49 × 10−7   0.19 × 10−7
propranolol   54 × 10−7   52 × 10−7
furosemide   u.d.l.a   u.d.l.a
a

Under detection limit.