Table 3.
PK parameters of intravenously administered DT3 or d6-DT3 (50 mg/Kg) in mice
Parameters | DT3 | d6-DT3 |
---|---|---|
AUC0-last (h·ng·mL−1) | 32804 | 34213 |
AUC0-∞ (h·ng·mL−1) | 33456 | 35707 |
Ke (h−1) | 0.0721 | 0.0656 |
Cl (L·Kg−1·h−1) | 1.495 | 1.400 |
Vd (L·Kg−1) | 20.7 | 21.3 |