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. Author manuscript; available in PMC: 2020 Sep 1.
Published in final edited form as: Curr Protoc Pharmacol. 2019 Sep;86(1):e67. doi: 10.1002/cpph.67

Table 1.

Recent natural product drug introductions, 2008-2018.

Year Drug name Company Indication NP template
2008 Biolimus stent Biosensors Stenosis Rapamycin
Ceftobiprole medocaril Roche Antibacterial Cephalosporin
Methyl naltrexone bromide Wyeth/Progenis Constipation Morphinan
2009 Nalfurafine HCl Toray Pruritis Morphinan
Tebipenem pivoxil Spero Antibacterial Thienamycin
Televancin Theravance Antibacterial Vancomycin
2010 Cabazitaxel Sanofi-Aventis Cancer Taxane
Ceftaroline fosamil Takeda Antibacterial Cephalosporin
Eribulin mesylate Eisai Cancer Halichondrin
Fingolimod Novartis Multiple sclerosis Myricocin
Mifamurtide Takeda Cancer Muramyl dipeptide
Romidepsin Fujisawa/Astellas Cancer Cyclopeptide
Vinflunine ditartate Pierre Fabre Cancer Vinca alkaloid
Zucapsaicin E Merck AG Topical analgesic Capsaicin
2011 Fidaxomicin Optimer Antibacterial Macrolide
Spinosad ParaPro Antiparasitic Spinosyn A
2012 Arterolane Ranbaxy Antiparasitic Artemisinin
Carfilzomib Proteolix.Onyx Cancer Peptide
Crofelemer Salix/Shaman Diarrhea Oligomeric proanthocyanin
Dapagliflozin Astra Zeneca Diabetes Phlorizin
Ingenol mebutate Peplin/Leo Cancer Phorbol ester
Novolimus Elixir Stenosis Rapamycin
Omacetaxine mepsuccinate ChemGenex/ Teva Cancer Homoharringtonine
Pixanthone dimaleate Cell Therapeutics Cancer Anthracycline
2013 Canagliflozin Jannsen Diabetes Phlorizin
2014 ---
2015 Ceftolozame Astellas/Cubist Antibacterial Cephalosporin
Dalbavancin Vicuron/Durata Antibacterial Vancomycin
Empagliflozin Boehringer/Lilly Diabetes Phlorizin
Nalogexol Nektar/Astra Zeneca Consitpation Morphinan
Oritavancin Lilly/Medicines Co. Antibacterial Vancomycin
Tofoglozin Chugai/Sanofi/Kowa Diabetes Phlorizin
2016 ---
2017 ---
2018 Midostaurin Novartis Cancer Staurosporine
Naldimedine Shionagi Constipation Morphinan