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. 2020 Aug 20;64(9):e00946-20. doi: 10.1128/AAC.00946-20

TABLE 4.

Papp value of SB-AF-1002 compared to those of cyclosporine and caffeine in monkey BBB kit

Drug Time (min) Papp (10−6 cm/s)
Cyclosporine 5 1
Cyclosporine 15 1
Cyclosporine 30 1
Caffeine 5 20
Caffeine 15 25
Caffeine 30 25
SB-AF-1002 5 6
SB-AF-1002 15 2
SB-AF-1002 30 1.1