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. 2020 Aug 18;25(16):3756. doi: 10.3390/molecules25163756

Table 2.

RT of stable gallium conjugates and [68Ga]Ga-radioconjugates of all aprepitant derivatives.

Stable Ga-Conjugate RT [68Ga]Ga-Radioconjugate RT
Ga-DOTA-Et-APT, Ga-5A 17.4 min [68Ga]Ga-DOTA-Et-APT, [68Ga]Ga-5A 17.7 min
Ga-DOTA-Pr-APT, Ga-5B 16.8 min [68Ga]Ga-DOTA-Pr-APT, [68Ga]Ga-5B 17.0 min
Ga-DOTA-Bu-APT, Ga-5C 16.9 min [68Ga]Ga-DOTA-Bu-APT, [68Ga]Ga-5C 17.3 min
Ga-DOTA-HN-NH-Ac-APT, Ga-5D 15.8 min [68Ga]Ga-DOTA-HN-NH-Ac-APT, [68Ga]Ga-5D 16.3 min
Ga-DOTA-Et-Ac-APT, Ga-5E 16.1 min [68Ga]Ga-DOTA-Et-Ac-APT, [68Ga]Ga-5E 16.5 min