Table 2.
Uptake of 211At Activity After Intravenous Administration of 211At-Labeled Murine 81C6 in Athymic Mice Bearing D54-MG Subcutaneous Xenografts
% Injected dose/grama |
||||
---|---|---|---|---|
Tissue | 2 h | 4 h | 16 h | 24 h |
Liver | 8.95 ± 1.91 | 9.55 ± 1.89 | 5.79 ± 2.28 | 5.62 ± 1.47 |
Spleen | 6.69 ± 1.12 | 7.83 ± 1.89 | 7.18 ± 1.87 | 7.30 ± 1.37 |
Lung | 14.94 ± 1.79 | 11.28 ± 2.09 | 11.17 ± 2.57 | 10.69 ± 1.52 |
Heart | 8.51 ± 1.98 | 7.00 ± 1.28 | 5.49 ± 1.43 | 5.42 ± 0.80 |
Kidney | 8.15 ± 0.58 | 7.12 ± 0.66 | 5.78 ± 1.03 | 5.70 ± 1.16 |
Stomach | 3.97 ± 0.48 | 6.60 ± 1.57 | 5.32 ± 0.60 | 8.15 ± 3.52 |
Sm. Int. | 2.82 ± 0.11 | 2.71 ± 0.20 | 2. 35 ± 0.43 | 2.86 ± 0.42 |
Lg. Int. | 1.39 ± 0.15 | 1.5 ± 0.25 | 1.46 ± 0.25 | 1.98 ± 0.35 |
Thyroidb | 1.18 ± 0.34 | 0.86 ± 0.35 | 0.56 ± 0.14 | 0.80 ± 0.25 |
Muscle | 0.96 ± 0.19 | 0.86 ± 0.20 | 0.98 ± 0.43 | 1.31 ± 0.21 |
Blood | 28.84 ± 1.93 | 21.11 ± 2.69 | 14.28 ± 3.11 | 15.65 ± 3.67 |
Bone | 3.10 ± 0.51 | 3.18 ± 0.57 | 3.22 ± 1.19 | 3.16 ± 0.53 |
Brain | 1.18 ± 0.26 | 0.79 ± 0.19 | 0.72 ± 0.16 | 0.75 ± 0.11 |
Tumor | 8.30 ± 1.72 | 10.78 ± 0.80 | 19.89 ± 2.97 | 19.40 ± 4.12 |
Mean ± SD (n = 5).
Injected dose per organ.