Table 5. Mouse Pharmacokinetic Profile of 7fa.
| dose (mg/kg) |
||
|---|---|---|
| 3 (IV) | 15 (PO) | |
| Tmax (h) | 0.5 | |
| Cmax (nM) | 1628 | |
| Cl (mL/min/kg) | 7.7 | |
| Vss (L/kg) | 20 | |
| T1/2 (h) | 32 | |
| F (%) | 62 | |
IV vehicle: 70/30 PEG400/water. PO vehicle: 80/20 PEG400/200 mM citrate buffer (pH 3.0).
| dose (mg/kg) |
||
|---|---|---|
| 3 (IV) | 15 (PO) | |
| Tmax (h) | 0.5 | |
| Cmax (nM) | 1628 | |
| Cl (mL/min/kg) | 7.7 | |
| Vss (L/kg) | 20 | |
| T1/2 (h) | 32 | |
| F (%) | 62 | |
IV vehicle: 70/30 PEG400/water. PO vehicle: 80/20 PEG400/200 mM citrate buffer (pH 3.0).