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. 2020 Jul 29;11(9):1751–1758. doi: 10.1021/acsmedchemlett.0c00264

Table 5. Mouse Pharmacokinetic Profile of 7fa.

  dose (mg/kg)
  3 (IV) 15 (PO)
Tmax (h)   0.5
Cmax (nM)   1628
Cl (mL/min/kg) 7.7  
Vss (L/kg) 20  
T1/2 (h) 32  
F (%)   62
a

IV vehicle: 70/30 PEG400/water. PO vehicle: 80/20 PEG400/200 mM citrate buffer (pH 3.0).