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. 2020 Apr 14;21(15):2111–2115. doi: 10.1002/cbic.202000117

Table 1.

IC50 [μM] values of ReI tricarbonyl complexes.8, 9, 13, 28

 

Complex

Cell line

V [a]

VI [b]

VII [b]

VIII [b]

IX [a]

KB‐3‐1

0.92±0.2

KBCP20

1.6±0.4

A2780

2.2±0.2

A2780CP70

3.0±0.7

A549

133.2±4.3

2.2±0.2

1.1±0.1

0.8±0.1

6.7±4.9

AF49CisR

2.1±0.1

8.3±0.1

2.1±0.1

5.4±1.8

H460

4.5±0.7

H460CisR

5.3±2.9

MRC‐5

4.1±0.9

HeLa

126.4±2.8

1.8±0.2

1.6±0.1

1.8±0.1

1.2±0.2

U2SO

1.4±0.1

1.1±0.1

MCF‐7

51.4±3.0

2.2±0.3

11.8±1.3

1.5±0.1

PC3

59.4±3.8

>25

1.1±0.1

HepG2

>25

1.6±0.1

LO2

7.5±0.1

2.0±0.1

HLF

12.7±0.8

MDA‐MB‐231

48.5±2.8

HT‐29

47.5±0.9

[a] 72 h incubation/MTT assay [b] 44 h incubation/MTT assay.