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. 2020 Mar 5;38(5):1570–1579. doi: 10.1007/s10637-020-00910-9

Table 2.

Drug-related TEAEs by CTC grade (≥10%)

Gal + TMZ/RTX (N = 40) TMZ/RTX (N = 16)
Grade 1–2 Grade ≥3 All Grade Grade 1–2 Grade ≥3 All Grade
Laboratory Event
 Platelet count decreased 12 (30.0) 6 (15.0) 18 (45) 3 (18.8) 1 (6.3) 4 (25.1)
 Lymphocyte count decreased 5 (12.5) 8 (20.0) 13 (32.5) 2 (12.5) 1 (6.3) 3 (18.8)
 White blood cells decreased 8 (20.0) 4 (10.0) 12 (30) 1 (6.3) 0 (0.0) 1 (6.3)
 ALT increased 4 (10.0) 3 (7.5) 7 (17.5) 2 (12.5) 0 (0.0) 2 (12.5)
 Neutrophil count decreased 5 (12.5) 2 (5.0) 7 (17.5) 2 (12.5) 0 (0.0) 2 (12.5)
 Anaemia 6 (15.0) 0 (0.0) 6 (15) 0 (0.0) 0 (0.0) 0 (0.0)
Non-laboratory Event
 Fatigue 24 (60.0) 1 (2.5) 25 (62.5) 6 (37.5) 0 (0.0) 6 (37.5)
 Nausea 21 (52.5) 0 (0.0) 21 (52.5) 8 (50.0) 1 (6.3) 9 (56.3)
 Constipation 16 (40.0) 0 (0.0) 16 (40) 4 (25.0) 0 (0.0) 4 (25.0)
 Alopecia 16 (40.0) 0 (0.0) 16 (40) 3 (18.8) 0 (0.0) 3 (18.8)
 Vomiting 11 (27.5) 1 (2.5) 12 (30) 5 (31.3) 0 (0.0) 5 (31.3)
 Decreased Appetite 8 (20.0) 0 (0.0) 8 (20) 2 (12.5) 0 (0.0) 2 (12.5)
 Headache 6 (15.0) 0 (0.0) 6 (15) 2 (12.5) 0 (0.0) 2 (12.5)
 Dyspepsia 5 (12.5) 0 (0.0) 5 (12.5) 1 (6.3) 0 (0.0) 1 (6.3)
 Weight decreased 5 (12.5) 0 (0.0) 5 (12.5) 1 (6.3) 0 (0.0) 1 (6.3)

To note: data given as No. (%) unless otherwise indicated

ALT alanine aminotransferase, Gal galunisertib, TMZ temozolomide, RTX radiation, TEAE treatment-emergent adverse events