SC |
Synthetic cannabinoid |
THC |
Tetrahydrocannabinol |
GIRK |
G protein-gated inward rectifier K+
|
SAR |
Structure versus activity relationship |
GPCR |
G protein-coupled receptor |
EMCDDA |
European Monitoring Centre for Drugs & Drug Addiction |
TRP |
Transient receptor potential |
ERK1/2 |
Extracellular signal-regulated kinase 1/2 |
AEA |
Anandamide |
2AG |
2-Arachidonoylglycerol |
EC50
|
Half-maximal effective concentration |
Emax
|
Maximal response |
FRET |
Förster resonance energy transfer |
CNG |
Cyclic nucleotide-gated |
BRET |
Bioluminescence resonance energy transfer |
MPSD |
Membrane potential-sensitive dye |
TM |
Transmembrane domains |