Table 5. In vivo antileishmanial activity against L. donovani in a golden hamster model.
| Compd. no | Percentage inhibition |
Route of administration | Dose mg kg–1 | |
| 7th day | 28th day | |||
| 1h | 36.0 ± 8.48 | NI | IP | 50 |
| 1k | 39.5 ± 0.70 | 29.0 ± 0.0 | IP | 50 |
| 1m | 36.0 ± 20.20 | 71.25 ± 10.56 | IP | 50 |
| 1m | 48.41 ± 11.44 | 66.03 ± 8.74 | Oral | 100 |
| 4bb | 44.02 ± 12.63 | 75.20 ± 6.64 | IP | 50 |
| 4kd | 29.22 ± 41.32 | NI | IP | 50 |
| 4kk | 50.92 ± 8.48 | 38.04 ± 2.6 | IP | 50 |
| 4md | 13.51 ± 0.6 | 2.08 ± 3.6 | IP | 50 |
| 4mf | 71.08 ± 11.11 | 28.63 ± 11.04 | IP | 50 |
| 4mf | 69.47 ± 8.34 | 12.70 ± 8.91 | Oral | 100 |
| 6ba | NI | NI | IP | 50 |
| 6gc | NI | NI | IP | 50 |
| 6ka | 19.32 ± 3.06 | NI | IP | 50 |
| 6kb | 61.99 ± 2.46 | 9.23 ± 6.12 | IP | 50 |
| 6mc | 20.01 ± 8.22 | 4.38 ± 5.28 | IP | 50 |
| Miltefosine | 97.32 ± 0.55 | 98.41 ± 1.41 | Oral | 30 |