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The binding affinity assay of compounds 24, 25, 26, 27, 28 and morphine on MOR.
| [3H]diprenorphine binding, Ki (nM) | |
|---|---|
| Morphine | 6 ± 1.0 |
| ME | 3.5 ± 0.8 |
| 24 | 830 ± 50.0 |
| 25 | 625 ± 79.0 |
| 26 | 535 ± 50.0 |
| 27 | 720 ± 95.0 |
| 28 | 965 ± 110.0 |
[Met5] Enkephalin (ME) is an opioid pentapeptide.
