Table 2. BCL-XL and BCL-2 TR-FRET Binding Data of THIQ-Pyridine Analogs 4–7.
| Compound | BCL-XL FRET Ki (nM) | BCL-2 FRET Ki (nM) |
|---|---|---|
| 4 | 11 | 626 |
| 5 | 0.329 | 119 |
| 6 | 0.296 | 117 |
| 7 | 5.96 | 348 |
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