TABLE 7.
Compound | EC50 (μM) | |||||||
---|---|---|---|---|---|---|---|---|
V370A | ΔV370 | Q369H | T371A | V362I | V370M | V370A/ΔT371 | ΔV371 | |
63 | 0.0025 | 0.014 | - | 0.0017 | 0.00094 | - | - | - |
64 | 0.0027 | 0.013 | 0.0019 | 0.002 | 0.0045 | 0.0028 | 0.0036 | 0.0073 |
-: Not determined
Compound | EC50 (μM) | |||||||
---|---|---|---|---|---|---|---|---|
V370A | ΔV370 | Q369H | T371A | V362I | V370M | V370A/ΔT371 | ΔV371 | |
63 | 0.0025 | 0.014 | - | 0.0017 | 0.00094 | - | - | - |
64 | 0.0027 | 0.013 | 0.0019 | 0.002 | 0.0045 | 0.0028 | 0.0036 | 0.0073 |
-: Not determined