Figure 1.

Development of DPAGT1 Inhibitors of Capuramycin Analogues. Structures of Capuramcyin, O-Methyl capuramycin (OM-Cap), Capuramycin phenoxypiperidinylbenzylamide analogue (CPPB), Aminouridyl phenoxylpiperidinylbenzylbutanamide (APPB, Previously Reported DPAGT1 Inhibitor), and Tunicamycin (Reference Molecule).