No. | R1 | R2 | R3 | X | No. | Yield (%) |
---|---|---|---|---|---|---|
5 | H | H | H | CH | 21 | 95 |
6 | H | H | Et | CH | 22 | 93 |
7 | Me | H | H | CH | 23 | 85 |
8 | Me | Me | H | CH | 24 | 88 |
9 | H | H | H | N | 25 | 88 |
10 | H | H | Et | N | 26 | 91 |
11 | Me | H | H | N | 27 | 87 |
12 | Me | Me | H | N | 28 | 64 |
No. | R1 | R2 | R3 | X | No. | Yield (%) |
---|---|---|---|---|---|---|
5 | H | H | H | CH | 21 | 95 |
6 | H | H | Et | CH | 22 | 93 |
7 | Me | H | H | CH | 23 | 85 |
8 | Me | Me | H | CH | 24 | 88 |
9 | H | H | H | N | 25 | 88 |
10 | H | H | Et | N | 26 | 91 |
11 | Me | H | H | N | 27 | 87 |
12 | Me | Me | H | N | 28 | 64 |