Table 4.
Compound | Relation | Value [mmol/L] | Standard | Microorganism Strain | Source |
---|---|---|---|---|---|
BA | >= | 0.52 | MIC | Staphylococcus aureus | [144] |
> | 1.05 | MIC | Staphylococcus aureus | [144] | |
= | 6.55 | MIC | Saccharomyces cerevisiae | [145] | |
= | 6.55 | MIC | Saccharomyces cerevisiae | [145] | |
= | 6.55 | MIC | Saccharomyces cerevisiae | [145] | |
= | 6.55 | MIC | Phellinus tremulae | [146] | |
> | 13.10 | MIC | Saccharomyces cerevisiae | [145] | |
> | 13.10 | MIC | Saccharomyces cerevisiae | [145] | |
= | 0.33 | MIC | Mycobacterium tuberculosis | [147] | |
= | 5.00 | MIC | Cochliobolus lunatus | [148] | |
= | 5.00 | MIC | Lasiodiplodia theobromae | [146] | |
= | 5.00 | MIC | Neofusicoccum ribis | [146] | |
= | 5.00 | MIC | Diplodia seriata | [146] | |
= | 5.00 | MIC | Botryosphaeria dothidea | [146] | |
CinA | = | 3.37 | MIC | Aspergillus parasiticus | [149] |
> | 0.86 | MIC | Streptococcus pyogenes | [150] | |
> | 0.86 | MIC | Staphylococcus aureus | [150] | |
= | 0.27 | MIC | Mycobacterium tuberculosis H37Rv | [151] | |
= | 1.68 | MIC | Aspergillus niger | [149] | |
= | 3.37 | MIC | Staphylococcus aureus | [149] | |
> | 0.86 | MIC | Staphylococcus epidermidis | [150] | |
= | 6.75 | MIC | Klebsiella pneumoniae | [149] | |
= | 6.75 | MIC | Bacillus subtilis | [149] | |
> | 0.86 | MIC | Pseudomonas aeruginosa | [150] | |
> | 0.86 | MIC | Staphylococcus aureus | [150] | |
= | 0.42 | MIC | Trichophyton rubrum | [149] | |
> | 0.86 | MIC | Escherichia coli | [150] | |
= | 0.84 | MIC | Issatchenkia orientalis | [149] | |
= | 6.75 | MIC | Burkholderia cepacia | [149] | |
= | 6.75 | MIC | Micrococcus luteus | [149] | |
= | 6.75 | MIC | Enterobacter cloacae | [149] | |
> | 0.86 | MIC | Bacillus subtilis | [150] | |
> | 0.60 | MIC | Mycobacterium smegmatis str. MC2 155 | [151] | |
= | 13.50 | MIC | Pseudomonas aeruginosa | [149] | |
p-CA | > | 0.60 | MIC | Mycobacterium smegmatis str. MC2 155 | [151] |
= | 5.00 | MIC | Diplodia seriata | [146] | |
> | 305 | MIC | Bacillus subtilis | [152] | |
= | 0.24 | MIC | Mycobacterium tuberculosis H37Rv | [151] | |
= | 5.00 | MIC | Neofusicoccum ribis | [146] | |
> | 305 | MIC | Candida albicans | [152] | |
> | 305 | MIC | Staphylococcus aureus | [152] | |
= | 5.00 | MIC | Botryosphaeria dothidea | [146] | |
> | 305 | MIC | Pseudomonas fluorescens | [152] | |
= | 0.37 | MIC | Mycobacterium bovis BCG | [151] | |
CFA | > | 0.28 | MIC | Bacillus subtilis | [152] |
> | 0.28 | MIC | Staphylococcus aureus | [152] | |
= | 0.71 | MIC50 | Candida albicans | [153] | |
= | 0.69 | MIC | Streptococcus pyogenes | [154] | |
= | 0.69 | MIC | Staphylococcus aureus | [154] | |
> | 0.30 | IC50 | Saccharomyces cerevisiae | [155] | |
> | 0.28 | MIC | Pseudomonas fluorescens | [152] | |
> | 0.35 | IC50 | Agaricus bisporus | [156] | |
= | 1.47 | MIC50 | Candida albicans | [153] | |
= | 0.28 | MIC50 | Candida albicans | [153] | |
> | 0.28 | MIC | Candida albicans | [152] | |
= | 0.71 | MIC50 | Candida albicans | [153] | |
RA | > | 5556 | MIC | Aspergillus niger | [157] |
= | 11111 | MIC | Aspergillus niger | [158] | |
= | 333 | MBC | Bacillus subtilis subsp. spizizenii | [157] | |
= | 11111 | MBC | Bacillus subtilis subsp. spizizenii | [158] | |
= | 11111 | MIC | Bacillus subtilis subsp. spizizenii | [158] | |
> | 5556 | MIC | Candida albicans | [157] | |
= | 5556 | MIC | Candida albicans | [158] | |
> | 5556 | MIC | Escherichia coli | [157] | |
= | 333 | MBC | Escherichia coli | [157] | |
> | 5556 | MIC | Pseudomonas aeruginosa | [157] | |
= | 333 | MBC | Pseudomonas aeruginosa | [157] | |
= | 11111 | MBC | Pseudomonas aeruginosa | [158] | |
= | 5556 | MIC | Pseudomonas aeruginosa | [158] | |
= | 333 | MIC | Staphylococcus aureus | [157] | |
= | 333 | MBC | Staphylococcus aureus | [157] | |
= | 333 | MBC | Staphylococcus aureus | [158] | |
= | 333 | MIC | Staphylococcus aureus | [158] | |
= | 333 | MIC | Staphylococcus epidermidis | [157] | |
= | 333 | MBC | Staphylococcus epidermidis | [157] | |
= | 2778 | MBC | Staphylococcus epidermidis | [158] | |
= | 333 | MIC | Staphylococcus epidermidis | [158] | |
D-ChA | = | 0.0039 | Ki | Clostridium botulinum * | [159] |
= | 0.0067 | Ki | Clostridium botulinum # | [159] | |
= | 0.0016 | Ki | Clostridium botulinum ** | [159] | |
= | 0.0014 | Ki | Clostridium botulinum ## | [159] | |
L-ChA | = | 0.0158 | Potency | Bacillus anthracis str. A2012 | [160] |
MIC—minimum inhibitory concentration, MIC50—minimum inhibitory concentration required to inhibit the growth of 50% of microorganisms, Ki—inhibitory constant, MBC—minimum bactericidal concentration, IC50—the half maximal inhibitory concentration. Uncompetitive inhibition of Clostridium botulinum: * full length BoNT/A light chain (1-448) using truncated SNAP 25 (141-206) peptide as substrate by LC/MS analysis, ** truncated BoNT/A light chain (1-425) using truncated SNAP 25 (141-206) peptide as substrate by LC/MS analysis, Competitive inhibition of Clostridium botulinum: # truncated BoNT/A light chain (1-425) using truncated SNAP 25 (141-206) peptide as substrate by LC/MS analysis, ## full length BoNT/A light chain (1-448) using truncated SNAP 25 (141-206) peptide as substrate by LC/MS analysis.