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. 2020 Oct 15;25(20):4724. doi: 10.3390/molecules25204724
A active
A2AR adenosine A2A receptor
APJR apelin receptor
AT1R angiotensin receptor 1
Azi p-azido-phenylalanine
β2AR β2 adrenergic receptor
B1/2R bradykinin receptor 1/2
BNPS-skatole 3-bromo-3-methyl-2-(2-nitrophenylthio)-3H-indole
Bpa p-benzoyl-phenylalanine
BRET bioluminescence resonance energy transfer
BTFA 3-bromo-1,1,1-trifluoroacetone
CCR5 CC chemokine receptor 5
CGRP calcitonin gene-related peptide
CRF corticopin-releasing factor
CRF1/2R corticopin-releasing factor receptor 1/2
CuAAC copper-catalyzed azide-alkyne cycloaddition
CXCL12 CXC chemokine ligand 12
CXCR4 CXC chemokine receptor 4
CPMG Carr-Purcell-Meiboom-Gill (pulse sequence)
cwEPR continuous wave EPR
DDM n-dodecyl-β-d-maltopyranoside
DEER double electron-electron resonance
ECD extracellular domain
ECL extracellular loop
EM electron microscopy
EPR electron paramagnetic resonance
ETB endothelin B receptor
FlAsH fluorescein arsenical hairpin binder
FRET fluorescence/Förster resonance energy transfer
FTIR Fourier-transform infrared spectroscopy
GLP-1 glucagon-like peptide-1
GLP1R glucagon-like peptide-1 receptor
GLR glucagon receptor
GPCR G protein-coupled receptor
HDX hydrogen-deuterium exchange
HRF hydroxyl radical footprinting
I inactive
LRET lanthanoid resonance energy transfer
MIP1α macrophage inflammatory protein 1α (=CCL3)
MS mass spectrometry
MTSL (1-oxyl-2,2,5,5-tetramethyl-pyrroline-3-methyl) methanethiosulfonate
ncAA non-canonical amino acid
NMR nuclear magnetic resonance
NOE nuclear Overhauser effect
NPY neuropeptide Y
NTS1R neurotensin receptor 1
PACAP pituitary adenylate cyclase-activating peptide
PAC1R pituitary adenylate cyclase-activating peptide receptor 1
PTH1R parathyroid hormone receptor 1
REDOR rotational-echo double-resonance
SAR structure activity relationship studies
SDS-PAGE sodium dodecyl sulfate–polyacrylamide gel electrophoresis
SDSL site-directed spin labeling
SPAAC strain-promoted azide-alkyne cycloaddition
STD saturation transfer difference spectroscopy
TCS transferred cross saturation spectroscopy
TET 2,2,2-trifluoro-ethanethiol
TM transmembrane
trNOESY transferred nuclear Overhauser effect spectroscopy
Uaa unnatural amino acid
Ucn Urocortin
Y1/2R neuropeptide Y receptor 1/2