Official websites use .gov
A
.gov website belongs to an official
government organization in the United States.
Secure .gov websites use HTTPS
A lock (
) or https:// means you've safely
connected to the .gov website. Share sensitive
information only on official, secure websites.
Inhibition potency of phosphoramidate inhibitors of PSMA
| Entry | IC50 (nM)a |
|---|---|
| 3 | 27 (3) |
| 4 | 19 (1) |
| 5 | 1.3 (0.08) |
| 6 | 0.4 (0.05) |
| 7a | 60 (11) |
| 7b | 357 (29) |
| 8a | 79 (6) |
| 8b | 112 (8) |
| 9a | 2.6 (0.2) |
| 9b | 3.0 (0.3) |
| 10a | 1.3 (0.2) |
| 10b | 11 (0.8) |
Standard deviation in parentheses.
