. 2020 Oct 10;21(20):7470. doi: 10.3390/ijms21207470

Table 2.

A1AR Modulators Trialed in Humans.

Receptor	Activity	Drug Acronym	Therapeutic Target (Reference)
A1AR	Agonist	SDZWAG994	Hypertriglyceridemia [88]
A1AR	Agonist	ARA	Hypertriglyceridemia [89]
A1AR	Agonist	RPR749	Hypertriglyceridemia [90]
A1AR	Partial agonist	GS-9667	Hyperlipidemia [91]