Skip to main content
. 2020 Sep 4;15(19):1776–1782. doi: 10.1002/cmdc.202000524

Figure 3.

Figure 3

Activity‐directed discovery of AR modulators by fragment growth. a) Structure of a fragment that binds to AR. b) Potential intermolecular reactions of the diazo substrates B14. c) Evolution of the structure of AR modulators through three rounds of ADS.