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. Author manuscript; available in PMC: 2025 Jan 1.
Published in final edited form as: Lancet Infect Dis. 2024 Sep 26;25(1):e47–e58. doi: 10.1016/S1473-3099(24)00512-7

Table 3. Characteristics of individual drugs for use in TBM.

Anti-TB
activity
Clinical
efficacy in TBM
Site of
disease exposure
Safety/
tolerability
Drug-drug
interactions
Access
Rifampicin 3 2 3 2 0 2
Isoniazid 3 2 3 2 1 2
Linezolid 74 2 2 3 1 1 2
Fluoroquinolones 50 3 2 3 2 1 2
Pyrazinamide 2 2 3 2 1 2
Pretomanid/delamanid 75 3 1 3 2 1 2
Bedaquiline 3 1 2 2 0 2
Alpibectir/ethionamide 2 0 3 2 1
Rifabutin 3 0 2 2 0 2
Clofazimine 1 0 1 2 1 2
Ethionamide 1 2 2 1 2
Cycloserine 1 0 2 1 2
Ethambutol 1 2 1 2
DprE1 inhibitors 3 0 0 2 1

Scores derived from the scoring system in Table 2.