Table 2. Summary of adverse events.
Standard of care in the abiraterone and enzalutamide trial (n=454) | Standard of care plus abiraterone and enzalutamide in the abiraterone and enzalutamide trial (n=445) | ||||||||
---|---|---|---|---|---|---|---|---|---|
Grade 1-2 | Grade 3 | Grade 4 | Grade 5 | Grade 1-2 | Grade 3 | Grade 4 | Grade 5 | ||
Blood and lymphatic | 193 (43%) | 21 (5%) | 5 (1%) | 0 | 217 (49%) | 9 (2%) | 4 (1%) | 0 | |
Cardiac | 25 (6%) | 10 (2%) | 5 (1%) | 0 | 45 (10%) | 19 (4%) | 7 (2%) | 5 (1%)* | |
Eye | 54 (12%) | 5 (1%) | 0 | 0 | 73 (16%) | 6 (1%) | 0 | 0 | |
Gastrointestinal and hepatobiliary | 242 (53%) | 19 (4%) | 4 (1%) | 1 (<1%) | 305 (69%) | 30 (7%) | 6 (1%) | 0 | |
General disorders and administration site conditions | 329 (72%) | 29 (6%) | 1 (<1%) | 0 | 348 (78%) | 54 (12%) | 2 (<1%) | 2 (<1%) | |
Fatigue | 296 (65%) | 13 (3%) | 0 | 0 | 348 (78%) | 34 (8%) | 0 | 0 | |
Infections | 89 (20%) | 17 (4%) | 1 (<1%) | 1 (<1%) | 101 (23%) | 22 (5%) | 3 (1%) | 3 (1%) | |
Injury | 8 (2%) | 6 (1%) | 0 | 0 | 23 (5%) | 11 (2%) | 0 | 0 | |
Investigations | 216 (48%) | 25 (6%) | 10 (2%) | 0 | 246 (55%) | 66 (15%) | 10 (2%) | 0 | |
Alanine aminotransferase increased | 75 (17%) | 3 (1%) | 0 | 0 | 112 (25%) | 44 (10%) | 1 (<1%) | 0 | |
Aspartate aminotransferase increased | 17 (4%) | 0 | 0 | 0 | 43 (10%) | 9 (2%) | 0 | 0 | |
Metabolism and nutrition | 143 (31%) | 6 (1%) | 0 | 0 | 190 (43%) | 17 (4%) | 3 (1%) | 0 | |
Glucose intolerance | 31 (7%) | 1 (<1%) | 0 | 0 | 23 (5%) | 7 (2%) | 0 | 0 | |
Hypokalaemia | 21 (5%) | 0 | 0 | 0 | 66 (15%) | 7 (2%) | 2 (<1%) | 0 | |
Musculoskeletal | 288 (63%) | 45 (10%) | 0 | 0 | 292 (66%) | 54 (12%) | 0 | 0 | |
Nervous system | 144 (32%) | 15 (3%) | 1 (<1%) | 0 | 232 (52%) | 20 (4%) | 6 (1%) | 0 | |
Seizure | 1 (<1%) | 0 | 0 | 0 | 0 | 4 (1%) | 0 | 0 | |
Cognitive disturbance | 22 (5%) | 2 (<1%) | 0 | 0 | 83 (19%) | 2 (<1%) | 1 (<1%) | 0 | |
Psychiatric | 187(41%) | 6 (1%) | 0 | 0 | 230 (52%) | 3 (1%) | 1 (<1%) | 0 | |
Renal and urinary | 292 (64%) | 17 (4%) | 5 (1%) | 0 | 306 (69%) | 18 (4%) | 5 (1%) | 2 (<1%) | |
Reproductive | 179 (39%) | 58 (13%) | 0 | 0 | 194 (44%) | 78 (18%) | 0 | 0 | |
Respiratory | 161 (35%) | 9 (2%) | 2 (<1%) | 0 | 196 (44%) | 12 (3%) | 1 (<1%) | 1 (<1%) | |
Skin | 121 (27%) | 4 (1%) | 1 (<1%) | 0 | 167 (38%) | 3 (1%) | 1 (<1%) | 0 | |
Vascular | 365 (80%) | 24 (5%) | 1 (<1%) | 0 | 324 (73%) | 93 (21%) | 1 (<1%) | 0 | |
Hypertension | 60 (13%) | 12 (3%) | 0 | 0 | 187 (42%) | 69 (16%) | 0 | 0 | |
Hot flushes | 365 (80%) | 12 (3%) | 0 | 0 | 374 (84%) | 24 (5%) | 0 | 0 |
Grade 1–2 adverse events occurring in 10% or more of patients in any treatment group or any grade 3, 4, or 5 adverse events stratified by body system, including adverse events of special interest. Abiraterone refers to abiraterone acetate and prednisolone. All adverse events in the abiraterone trial are shown in the appendix (p 7). *Events on old form categorised as “Cardiovascular—other” have been included in the cardiac body system.