Table 2.
IC50 values determined from fits of pinacidil concentration-response relationships (using Hill equation) for popliteal lymphatics from WT, Kir6.1−/− and SUR2[STOP] mice.
Parameter | WT | Kir6.1−/− | SUR2[STOP] |
---|---|---|---|
Normalized AMP IC50 (M) | 3.4 ·10−7 | 1.4 ·10−4 | 7.0 ·10−4 |
Normalized FREQ IC50 (M) | 1.3 ·10−7 | 8.3 ·10−5 | 4.1 ·10−4 |
Change in Tone IC50 (M) | n/a | n/a | n/a |
All parameters were normalized to those averaged over the 2-min period prior to administration of the first pinacidil dose. M = molar. n/a = could not be fit to Hill equation.