Table 4.

Effect of compounds 2–17 on HIV-1 RDDP and IN functions.

Compound	IC50 (µM)
	RDDP	IN
2	>100	4.3 ± 1.5
3	60 ± 9	2.35 ± 0.44
4	57 ± 3	8.5 ± 0.3
5	>100	6.5 ± 2.5
6	63 ± 11	89 ± 10
7	23.4 ± 0.5	31.5 ± 6.5
8	26.7 ± 2.2	3.4 ± 0.83
9	46 ± 3	7 ± 2
10	30.5 ± 0.4	3.4 ± 0.6
11	>100	7.2 ± 0.7
12	>100	6.61 ± 0.93
13	99 ± 1	23.18 ± 0.8
14	>100	>100
15	25.3 ± 6.3	5.35 ± 0.35
16	38 ± 4	0.69 ± 0.19
17	70 ± 1	1.44 ± 0.40
EFV	0.010 ± 0.005	ND
RAL	ND	0.055 ± 0.002