Table 7. Mouse efficacy model of VL for 48 and 50.
Compound | Dosing regimen | % Suppression of parasite load |
48 | 30 mg kg–1b.i.d. for 5 days PO | 60 |
48 | 100 mg kg–1b.i.d. for 5 days PO | 98 |
50 | 25 mg kg–1b.i.d. for 5 days PO | 17 |
50 | 50 mg kg–1b.i.d. for 5 days PO | 57 |