| API | Active Pharmaceutical Ingredient |
| AUC | Area Under the Curve |
| CMC | Critical Micellar Concentration |
| CTAB | Cetyltrimethylammonium Bromide |
| CYP450 | Cytochrome P450 |
| DHB | Dihydroxybergamottin |
| DMSO | Dimethyl Sulfoxide |
| FA | Fatty Acids |
| GIT | Gastrointestinal Tract |
| HPC | Hydroxypropyl Cellulose |
| HPMC | Hydroxypropyl Methylcellulose |
| IC50 | Inhibitory Concentration |
| Ki | Inhibitory Constant |
| Clint | Intrinsic Clearance |
| mRNA | Messenger RNA |
| MDZ | Midazolam |
| Mw | Molecular weight |
| MDR1 | Multi-drug Resistance Gene |
| mPEGx-PCLx | Methoxy Poly(ethylene glycol)-poly(ε-caprolactone) (mPEGx-PCLx) |
| ATBC | Acetyl Tributyl Citrate |
| F68 | Pluronic F68 |
| PEG | Polyethylene Glycol |
| PVA | Polyvinyl Acetate |
| PVP | Polyvinyl Pyrrolidone |
| PXR | Pregnane X receptor |
| SDS | Sodium Dodecyl Sulfate |
| SEDSS | Self-emulsifying Drug Delivery System |
| SMEDDS | Self-micro Emulsifying Drug Delivery System |
| NaCMC | Sodium Carboxymethyl Cellulose |
| NI | No Inhibition |
| TPGS | D -α-Tocopherol Polyethylene Glycol 1000 Succinate |
| TX-100 | Triton X-100 |