| AChE | Acetylcholinesterase |
| AhR | Aryl hydrocarbon receptor |
| CAR | Constitutive androstane receptor |
| CYP | Cytochrome p450 |
| DDI | Drug–drug interaction |
| DME | Drug-metabolizing enzyme |
| NR | Nuclear receptor |
| OOTC | Organ-on-a-chip |
| PXR | Pregnane X receptor |
| qHTS | Quantitative high-throughput screening |
| UGT | Glucuronosyltransferase |
| 2D | Two dimensional |
| 3D | Three dimensional |