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. 2020 Sep 1;11(11):2131–2138. doi: 10.1021/acsmedchemlett.0c00272

Table 1. Binding of Series 1 Ligands to FBD35 and FKBP12.

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a

Determined by fluorescence polarization and fitting the data to a competitive inhibition model (nM).

b

Determined by differential scanning calorimetry (°C).

*

Incomplete displacement of fluorescent probe.