TABLE 1.
Reported activity of various β-lactamase inhibitors from the BLBLIs against β-lactamase enzymes
| Enzyme | Inhibited by: |
|||
|---|---|---|---|---|
| Avibactam | Tazobactam | Vaborbactam | Relebactam | |
| Class A | ||||
| KPC | Yes | No | Yes | Yes |
| SHV | Yes | Yes | Yes | Yes |
| TEM | Yes | Yes | Yes | Yes |
| CTX-M | Yes | Yes | Yes | Yes |
| Class B | ||||
| MBL | No | No | No | No |
| Class C | ||||
| AmpC | Yes | No | Yes | Yes |
| Class D | ||||
| OXA | VDa | No | No | VD |
VD, variable data.