Table 1. Human KOR Agonist in Vitro Activitya.
EC50 values are means of two or more runs with CR845 as positive control for each batch (CR845 KOR EC50 = 2.62 ± 0.75 pM, n = 5).
EC50 values are means of two or more runs with CR845 as positive control for each batch (CR845 KOR EC50 = 2.62 ± 0.75 pM, n = 5).