Skip to main content
. 2020 Sep 14;11(11):2151–2155. doi: 10.1021/acsmedchemlett.0c00287

Table 2. In Vitro Potency of SHR0687a.

Compound ID SHR0687
MW/AlogP/PSA 720.9/2.06/186.8
hKOR EC50 (pM) 0.53
hMOR EC50 (nM) >50000
hDOR EC50 (nM) >50000
a

The positive control for hMOR and hDOR test was morphine (hMOR EC50 = 79.12 ± 9.91 nM, n = 3; hDOR EC50 = 203.97 ± 33.51 nM, n = 3).