Table 2. In Vitro Potency of SHR0687a.
Compound ID | SHR0687 |
---|---|
MW/AlogP/PSA | 720.9/2.06/186.8 |
hKOR EC50 (pM) | 0.53 |
hMOR EC50 (nM) | >50000 |
hDOR EC50 (nM) | >50000 |
The positive control for hMOR and hDOR test was morphine (hMOR EC50 = 79.12 ± 9.91 nM, n = 3; hDOR EC50 = 203.97 ± 33.51 nM, n = 3).