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. 2020 Sep 24;11(11):2244–2252. doi: 10.1021/acsmedchemlett.0c00387

Table 5. Further Characterization and SAR of C3 Benzoic Acid and Phenylacetic Acid Azaindole Derivatives.

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a

Enzymatic kinase activity assay.

b

Ratio of PI3Kα or PI3Kδ enzymatic inhibition over PI3Kγ inhibition.

c

Cellular potency in THP-1 cell line.

d

Compound was tested once.

e

n.d. = value not determined.