Table 1.

Inhibition of CDD-97 and CDD-97 derivatives for structure-activity relationship studies (modified portion of derivatives is in bold).

Compound I.D.	Structure	Ki (μM)
6		> 50
7		0.76 ± 0.03
8		1.7 ± 0.3
9		2.2 ± 0.2
10		18.8 ± 2.5
11		7.8 ± 0.1
12		0.84 ± 0.03
13		0.61 ± 0.02
14		> 50
15		29 ± 4
16		0.26 ± 0.04