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. 2020 Jul 13;45(6):809–815. doi: 10.1007/s13318-020-00634-4
Citrus polymethoxyflavones and flavone rutinosides inhibit OATP2B1, and the polymethoxyflavones also inhibit OATP1B1 and OATP1B3.
Ingestion of these compounds might lead to interactions with OATP substrates.
Caution is recommended when using these compounds as a functional food or medicine.