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. 2020 Nov 23;37(12):249. doi: 10.1007/s11095-020-02955-0

Table V.

Binary PC-SAFT interaction parameters between excipients and APIs

FFB IBU IND CBZ GRI
kij, int
[−]
kij, slope
[T−1]
kij, int
[−]
kij, slope
[T−1]
kij, int
[−]
kij, slope
[T−1]
kij, int
[−]
kij, slope
[T−1]
kij, int
[−]
kij, slope
[T−1]
TG808080 −0.107 [9] 0.00030 −0.1370 [9] 0.00040 0.024 [9] 0 0.175 * 0 0.031 * 0
DG100100 −0.032 * 0 0.028 * 0 −0.013 * 0 0.040 * 0 0.020 * 0
MG80 −0.032 * 0 0.028 * 0 −0.013 * 0 0.040 * 0 0.020 * 0
MC80 −0.113 * 0.00028 0.027 * 0 0.008 * 0 0.028 * 0 0.028 * 0
Lauroglycol FCC −0.038 * 0 0.007 * 0 0.011 * 0 0.097 * 0 0.039 * 0
Capryol 90 −0.034 * 0 0.003 * 0 0.003 * 0 0.064 * 0 0.025 * 0
TPGS1000 −0.030 * 0 0.006 * 0 −0.014 * 0 0.023 * 0 −0.007 * 0
carbitol −0.013 * 0 0 0 −0.009 * 0 0.029 * 0 0.018 * 0
PEG400 0.028 * 0 0 0 0.004 * 0 −0.012 * 0 0.011 * 0
ethanol 0.033 [9] 0 0.1458 * −0.00030 0.0309 [33] −0.00008 0.079 [34] −0.00015 0.032 * 0
GLI NAP CIN PZQ FEL

kij, int

[−]

kij, slope

[T−1]

kij, int

[−]

kij, slope

[T−1]

kij, int

[−]

kij, slope

[T−1]

kij, int

[−]

kij, slope

[T−1]

kij, int

[−]

kij, slope

[T−1]

TG808080 0.024 * 0 0.041 * 0 0.026 * 0 0.017 * 0 0.007 * 0
DG100100 0.010 * 0 0.008 * 0 −0.006 * 0 −0.039 * 0 0.000 * 0
MG80 0.010 * 0 0.008 * 0 −0.006 * 0 −0.039 * 0 0.000 * 0
MC80 0.033 * 0 0.018 * 0 −0.034 * 0 0.000 * 0 0.024 * 0
Lauroglycol FCC 0.044 * 0 0.034 [17] 0 0.026 * 0 0.005 * 0 0.019 * 0
Capryol 90 0.023 * 0 0.013 [17] 0 0.019 * 0 0.007 * 0 0.005 * 0
TPGS1000 −0.011 * 0 −0.003 [17] 0 0.005 * 0 0.023 * 0 −0.016 * 0
carbitol 0.008 * 0 −0.011 * 0 0.006 * 0 0.014 * 0 0.003 * 0
PEG400 0.000 * 0 −0.017 * 0 0.010 * 0 0.058 * 0 0.011 * 0
ethanol −0.024 [35] 0.00013 −0.001 [33] 0 0.004 * 0 0.020 * 0 0.002 * 0

*The supporting experimental data can be obtained on request