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. Author manuscript; available in PMC: 2021 Jun 26.
Published in final edited form as: J Nat Prod. 2020 Jun 8;83(6):2010–2024. doi: 10.1021/acs.jnatprod.0c00404

Table 5.

GI50 Values for Compounds 1–10.a

compound cell line
MDA-MB-453 SUM-185PE MDA-MB-231
1 5.4 ± 0.9 3.9 ± 0.8 >100
2 3.5 ± 0.4 2.1 ± 0.8 >100
3 3.3 ± 2.2 2.1 ± 0.5 >100
4 3.7 ± 0.3 2.8 ± 0.6 >100
5 3.6 ± 0.5 8.0 ± 5.1 >100
6 2.5 ± 0.6 1.5 ± 0.1 >100
7 4.0 ± 0.7 2.2 ± 0.7 >100
8 7.9 ± 1.4 4.4 ± 0.7 >100
9 2.6 ± 0.6 2.0 ± 0.2 >100
10 2.3 ± 0.3 1.4 ± 0.2 >100
Rapamycin 0.05 ± 0.04 0.04 ± 0.01 >100
a

Concentrations (nM) that inhibit growth by 50%, n = 3 ± SD.