Table 2.

Chemical structure, CA IX inhibitory activity, CA I/ CA IX selectivity profile of the best compound for each class of CA glycoconjugated inhibitors

Class	Structure	Ki CA IX (nM)	Selectivity ratio CA I/ CA IX	Ref.
Topiramate derivatives		10	1070	28
Anomeric sulfamates		2	4750	29
S-glycosyl derivatives		94	72	31
Thioureido derivatives		2	2029	32
Amidophenyl sulfonamides		700	17.4	33
Glycosyl triazoles		6	60	47
Coumarin derivatives		9	>11	55
C-glycosyl derivatives		16	4	66