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. Author manuscript; available in PMC: 2020 Dec 29.
Published in final edited form as: J Med Chem. 2017 Jan 3;60(1):157–169. doi: 10.1021/acs.jmedchem.6b00923

Table 3.

PAMPA Results of 1–4

compd %T ± SD Papp ± SD (cm·s−1, × 10−6)
1 32.3 ± 2 14.3 ± 1.6
2 0.3 ± 0.08 0.08 ± 0.02
3 0.2 ± 0.04 0.13 ± 0.01
4 0.1 ± 0.09 0.04 ± 0.02