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. Author manuscript; available in PMC: 2021 Jan 6.
Published in final edited form as: J Med Chem. 2018 Mar 29;61(7):2989–3007. doi: 10.1021/acs.jmedchem.8b00068

Table 1.

Selectivities of 29 and 30 between β-Catenin/BCL9 over β-Catenin/E-Cadherin Interactionsa

Ki ± SD (μM)
compd β-catenin/BCL9 β-catenin/E-cadherin selectivity of BCL9/cadherin
29 0.47 ± 0.14 >915 >1900
30   1.6 ± 0.23 >915   >570
a

Each set of data was expressed as mean ± standard deviation (n = 3).