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. 2020 Dec 22;22(1):22. doi: 10.3390/ijms22010022

Table 1.

Trospium transport kinetics in man and mouse.

Human Carrier Km (µM) Vmax
(pmol/mg protein/min)
Mouse Carrier Km (µM) Vmax (pmol/mg protein/min)
OCT1 17 ± 5 [8] 93 ± 26 [8] mOct1 58.7 ± 15.5 352.9 ± 39.4
106 ± 16 [9] 269 ± 18 [9]
15 ± 3 [10] 1142 ± 157 [10]
OCT2 8 ± 1 [8] 92 ± 11 [8] mOct2 78.5 ± 25.9 899.3 ± 139.7
0.6 ± 0.1 [10] 98 ± 22 [10]
MATE1 15 ± 2 [10] 1083 ± 143 [10] mMate1 29.3 ± 6.7 184.7 ± 14.0
MATE2-K 8 ± 2 [10] 297 ± 6 [10] mMate2 No transport No transport