Table 1.
Trospium transport kinetics in man and mouse.
Human Carrier | Km (µM) | Vmax (pmol/mg protein/min) |
Mouse Carrier | Km (µM) | Vmax (pmol/mg protein/min) |
---|---|---|---|---|---|
OCT1 | 17 ± 5 [8] | 93 ± 26 [8] | mOct1 | 58.7 ± 15.5 | 352.9 ± 39.4 |
106 ± 16 [9] | 269 ± 18 [9] | ||||
15 ± 3 [10] | 1142 ± 157 [10] | ||||
OCT2 | 8 ± 1 [8] | 92 ± 11 [8] | mOct2 | 78.5 ± 25.9 | 899.3 ± 139.7 |
0.6 ± 0.1 [10] | 98 ± 22 [10] | ||||
MATE1 | 15 ± 2 [10] | 1083 ± 143 [10] | mMate1 | 29.3 ± 6.7 | 184.7 ± 14.0 |
MATE2-K | 8 ± 2 [10] | 297 ± 6 [10] | mMate2 | No transport | No transport |