Table 1. IC50a and pIC50 Values for Various 4-(Quinolin-5-yl)butanoic Amide Analogues.
IC50 values were taken as dose-dependent decreases in the EC80 acetylcholine response determined in CHO-K1 cells expressing the hM1R.
IC50 values were taken as dose-dependent decreases in the EC80 acetylcholine response determined in CHO-K1 cells expressing the hM1R.