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. 2021 Jan 4;64(1):719–740. doi: 10.1021/acs.jmedchem.0c01727

Table 8. Cross-Screening against mmpL3 Mutantsa.

strain 1 2 12 15 47 40 38
H37Rv WT MIC (μM) 1.7 4.8 15 27 5.8 1.2 1.2
MmpL3 F255L MIC (μM) 18 55 170 >200 41 >200 39
MmpL3 F644L MIC (μM) 1.9 5.4 17 24 5.5 1 1.9
MmpL3 V681 MIC (μM) 16 45   >200      
MmpL3 G596R MIC (μM) 40 110   >200      
a

WT: wild-type.