Table 8. Cross-Screening against mmpL3 Mutantsa.
strain | 1 | 2 | 12 | 15 | 47 | 40 | 38 |
---|---|---|---|---|---|---|---|
H37Rv WT MIC (μM) | 1.7 | 4.8 | 15 | 27 | 5.8 | 1.2 | 1.2 |
MmpL3 F255L MIC (μM) | 18 | 55 | 170 | >200 | 41 | >200 | 39 |
MmpL3 F644L MIC (μM) | 1.9 | 5.4 | 17 | 24 | 5.5 | 1 | 1.9 |
MmpL3 V681 MIC (μM) | 16 | 45 | >200 | ||||
MmpL3 G596R MIC (μM) | 40 | 110 | >200 |
WT: wild-type.