| A | Acidic |
| ACE(I) | angiotensin-converting enzyme (inhibitors) |
| AchRs | acetylcholine receptors |
| AIDS | acquired immune deficiency syndrome |
| Alloc | allyloxycarbonyl |
| AMPs | antimicrobial peptides |
| APCs | antigen presenting cells |
| APL | altered peptide ligands |
| ARB | angiotensin receptor blockers |
| B | basic |
| BAP | bioactive peptides |
| BOC | butoxycarbonyl |
| Bzl | benzyl |
| CG | coarse grain |
| COVID-19 | coronavirus disease 2019 |
| CPPs | cell penetrating peptides |
| CSD | Cambridge Structure Database |
| CTL | cytotoxic T lymphocyte |
| 2D | two-dimensional |
| 3D | three-dimensional |
| DH | degree of hydrolysis |
| DKP | diketopiperazines |
| DNA | deoxyribonucleic acid |
| EDTA | ethylenediaminetetraacetic acid |
| FAS | fatty acid synthase |
| FDA | Food and Drug Administration |
| FMOC | fluorenylmethoxycarbonyl |
| GALA | glutamic acid–alanine–leucine–alanine |
| GAS | group A streptococcus |
| GDS | gene delivery system |
| GFR | growth factor receptors |
| HeLa | human cervical cancer cell line |
| HIV | human immunodeficiency virus |
| HMG | high motility group |
| HMGR | 3-hydroxy-3-methylglutaryl CoA reductase |
| HOAt | 1-hydroxy-7-aza-benzotriazole |
| HOBt | 1-hydroxy-benzotriazole |
| HPLC | high performance liquid chromatography |
| IFN | interferon |
| IUPAC | International Union of Pure and Applied Chemistry |
| LDL | low-density lipoprotein |
| LDLR | LDL receptor |
| LF | lactoferrin |
| LPS | lipopolysaccharide |
| LRPs | low density lipoprotein receptors |
| LRs | leptin receptors |
| MBP | myelin basic protein |
| MD | molecular dynamics |
| MHC | major histocompatibility complex |
| NF | nuclear factor |
| NLSs | nuclear localization signals |
| NPC | nuclear pore complex |
| PDC | pyruvate dehydrogenase complexes |
| PEG | polyethylene glycol |
| PES | potential energy surface |
| PPI | proton-pump inhibitors |
| RAS | renin-angiotensin system |
| RCSB PDB | Research Collaboratory for Structural Bioinformatics Protein Data Bank |
| RGD | arginine–glycine–aspartic acid |
| RNA | ribonucleic acid |
| SARS-COV-2 | Severe Acute Respiratory Syndrome Coronavirus |
| SPPS | solid-phase synthesis |
| SREBP2 | sterol regulatory element-binding protein 2 |
| SWOT | strengths, weaknesses, opportunities, and threats |
| tBu | tert-butyl |
| TFA | trifluoroacetic acid |
| TFRs | transferrin receptors |
| TMC | trimethyl chitosan |
| TNF | tumor necrosis factor alpha |
| TNFR | tumor necrosis factor receptor 1 |