TABLE 1.
Tissues concentration (ng/g) and Kp_tissue/blood ratio of HCQ (mean ± SD).
Thymus (ng/g) | Kidney (ng/g) | Spleen (ng/g) | Liver (ng/g) | Heart (ng/g) | Subcutaneous Fat (ng/g) | Brain (ng/g) | Lung (ng/g) | BALF (ng/mL) | |
Group E: tissue concentration | 481.33 ± 242.24 | 79.70 ± 15.31 | 82.30 ± 34.37 | 78.83 ± 28.77 | 65.23 ± 21.37 | 35.22 ± 35.22 | 33.10 ± 11.46 | 20.77 ± 8.57 | 26.83 ± 11.19 |
Group E: Kp ratio | 223.25 ± 23.79 | 43.33 ± 22.42 | 39.91 ± 13.85 | 38.63 ± 11.25 | 32.16 ± 7.80 | 20.68 ± 25.51 | 16.40 ± 5.19 | 9.98 ± 2.09 | 1.33 ± 0.63 |
Group F: tissue concentration | 1,375.00 ± 219.20 | 1,115.00 ± 7.07 | 1,610.00 ± 1,032.38 | 3,025.00 ± 1,435.43 | 579.50 ± 120.92 | 75.55 ± 4.74 | 59.85 ± 11.81 | 738.50 ± 256.68 | 168.50 ± 40.31 |
Group F: Kp ratio | 11.54 ± 6.52 | 9.07 ± 3.90 | 11.29 ± 2.83 | 22.09 ± 1.22 | 4.91 ± 2.98 | 0.61 ± 0.22 | 0.47 ± 0.11 | 5.55 ± 0.46 | 0.13 ± 0.03 |