Table 1.
The AUCplasma, AUCbrain and z values of probe compounds following oral administration to WT and APP/PS1 mice. Data are presented as mean ± SD (n=3).
Compound | AUCplasma (ng·h/mL) | AUCbrain (ng·h/g) | ||||
---|---|---|---|---|---|---|
WT | APP/PS1 | z value | WT | APP/PS1 | z value | |
Caffeine | 10380 ± 738 | 11289 ± 681 | 0.90 | 21520 ± 224 | 22178 ± 356 | 1.56 |
Diazepam | 356.6 ± 35.6 | 343.3 ± 29.2 | 0.29 | 119.5 ± 5.5 | 117.7 ± 18.2 | 0.10 |
Valsartan | 1960 ± 231 | 1388 ± 105 | 2.26* | NA | NA | |
Digoxin | 199.4 ± 12.7 | 154.1 ± 16.8 | 2.14* | NA | NA |
NA: AUC value was not able to be calculated due to the detection limit of the brain assay.
z > 1.96 indicates a significant difference in AUCplasma or AUCbrain between WT and APP/PS1 mice.